|
SELECTED
PUBLICATIONS:
- A practical approach for repositioning
flipped venous access ports.
J Vasc Interv Radiol. 2000 Feb;11(2 Pt 1):213-4. No abstract
available.
PMID: 10716392 [PubMed - indexed for MEDLINE]
-
- Conformationally restricted analogs of
BD1008 and an antisense oligodeoxynucleotide targeting sigma1
receptors produce anti-cocaine effects in mice.
Eur J Pharmacol. 2001 May 11;419(2-3):163-74.
PMID: 11426838 [PubMed - indexed for MEDLINE]
-
- Synthesis and transporter binding
properties of bridged piperazine analogues of
1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR
12909).
J Med Chem. 2000 Dec 14;43(25):4840-9.
PMID: 11123994 [PubMed - indexed for MEDLINE]
-
| 4: |
Matecka
D, Rothman RB, Radesca L, de Costa BR, Dersch CM, Partilla JS,
Pert A, Glowa JR, Wojnicki FH, Rice KC. |
Related
Articles,
Links |
- Development of novel, potent, and
selective dopamine reuptake inhibitors through alteration of the
piperazine ring of 1-[2-(diphenylmethoxy)ethyl]-and
1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazines
(GBR 12935 and GBR 12909).
J Med Chem. 1996 Nov 22;39(24):4704-16.
PMID: 8941383 [PubMed - indexed for MEDLINE]
-
- Synthesis of N,N'-substituted piperazine
and homopiperazine derivatives with polyamine-like actions at
N-methyl-D-aspartate receptors.
J Med Chem. 1995 Dec 8;38(25):4891-6.
PMID: 8523402 [PubMed - indexed for MEDLINE]
-
- Characterization of two novel sigma
receptor ligands: antidystonic effects in rats suggest sigma receptor
antagonism.
Eur J Pharmacol. 1995 Jul 14;280(3):301-10.
PMID: 8566098 [PubMed - indexed for MEDLINE]
-
- A new approach to the design of
sigma-2-selective ligands: synthesis and evaluation of
N-[2-(3,4-dichlorophenyl)ethyl]-N-methyl-2-(1- pyrrolidinyl)ethylamine-related
polyamines at sigma-1 and sigma-2 receptor subtypes.
J Med Chem. 1994 Jan 21;37(2):314-21.
PMID: 8295220 [PubMed - indexed for MEDLINE]
-
- Further studies of the
structure-activity relationships of
1-[1-(2-benzo[b]thienyl)cyclohexyl]piperidine. Synthesis and
evaluation of 1-(2-benzo[b]thienyl)-N,N-dialkylcyclohexylamines at
dopamine uptake and phencyclidine binding sites.
J Med Chem. 1993 Dec 10;36(25):4075-81.
PMID: 8258830 [PubMed - indexed for MEDLINE]
-
- Synthesis, configuration, and activity
of isomeric 2-phenyl-2-(N-piperidinyl)bicyclo[3.1.0]hexanes at
phencyclidine and sigma binding sites.
J Med Chem. 1992 Dec 11;35(25):4704-12.
PMID: 1469699 [PubMed - indexed for MEDLINE]
-
- Synthesis and biological evaluation of
conformationally restricted
2-(1-pyrrolidinyl)-N-[2-(3,4-dichlorophenyl)ethyl]-N-methylethylenediam
ines as sigma receptor ligands. 1. Pyrrolidine, piperidine,
homopiperidine, and tetrahydroisoquinoline classes.
J Med Chem. 1992 Nov 13;35(23):4334-43.
PMID: 1447735 [PubMed - indexed for MEDLINE]
-
- Probes for narcotic receptor mediated
phenomena. 18. Epimeric 6 alpha- and 6
beta-iodo-3,14-dihydroxy-17-(cyclopropylmethyl)-4,5 alpha-epoxymorphinans
as potential ligands for opioid receptor single photon emission
computed tomography: synthesis, evaluation, and radiochemistry of
[125I]-6 beta-iodo-3,14-dihydroxy-17-(cyclopropylmethyl)-4,5 alpha-epoxymorphinan.
J Med Chem. 1992 Jul 24;35(15):2826-35.
PMID: 1322988 [PubMed - indexed for MEDLINE]
-
- Novel site-directed affinity ligands for
GABA-gated chloride channels: synthesis, characterization, and
molecular modeling of
1-(isothiocyanatophenyl)-4-tert-butyl-2,6,7-trioxabicyclo[2.2.2]octanes
.
J Med Chem. 1991 May;34(5):1531-8.
PMID: 2033577 [PubMed - indexed for MEDLINE]
-
- Characterization of benzodiazepine
receptors with a fluorescence-quenching ligand.
J Biol Chem. 1990 Dec 25;265(36):22181-6.
PMID: 2176206 [PubMed - indexed for MEDLINE]
-
| 14: |
de
Costa BR, Rice KC, Bowen WD, Thurkauf A, Rothman RB, Band L,
Jacobson AE, Radesca L, Contreras PC, Gray NM, et al. |
Related
Articles,
Links |
- Synthesis and evaluation of
N-substituted cis-N-methyl-2-(1-pyrrolidinyl)cyclohexylamines as high
affinity sigma receptor ligands. Identification of a new class of
highly potent and selective sigma receptor probes.
J Med Chem. 1990 Nov;33(11):3100-10.
PMID: 2172538 [PubMed - indexed for MEDLINE]
-
- Cannabinoid receptor localization in
brain.
Proc Natl Acad Sci U S A. 1990 Mar;87(5):1932-6.
PMID: 2308954 [PubMed - indexed for MEDLINE]
-
- Sunlight regulates the cutaneous
production of vitamin D3 by causing its photodegradation.
J Clin Endocrinol Metab. 1989 May;68(5):882-7.
PMID: 2541158 [PubMed - indexed for MEDLINE]
-
- Location of conjugated diene position in
an aliphatic chain by mass spectrometry of the
4-phenyl-1,2,4-triazoline-3,5-dione adduct.
Anal Chem. 1987 Aug 1;59(15):1954-7. No abstract available.
PMID: 3631517 [PubMed - indexed for MEDLINE]
-
-
BOOK CHAPTERS:
1:
Walker, J. M., Bowen, W. D., Walker, F. O., Matsumoto, R. R., de
Costa, B., and Rice, K. C.: Sigma Receptors:
Biology
and Function. Pharmacol. Rev.,
1990, 542,
355-402.
2:
de
Costa, B. R. and He, X.-S.: Synthesis, Structure-Activity Relationships
and Evolution of Sigma Receptor Ligands (1976-Present).
Neuroscience Perspectives Series. Itzhak, J. and Chapman, C.: Eds.:
Academic Press,1993, 45-111.
e-mail: briandecosta@charter.net
|
